Basic Information
ID: ALA5216204
Type: Binding
Description: Inhibition of PI3K p110alpha/p85alpha (unknown origin) using PIP2 as substrate preincubated for 15 mins followed by substrate addition measured after 1 hr in presence of ATP by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5216204
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 507.45 | 3.00 | 3.00 |
| 441.52 | 2.30 | 2.30 |
| 435.49 | 2.15 | 2.15 |
| 427.51 | 1.38 | 1.38 |
| 463.47 | 2.88 | 2.88 |
| 455.54 | 2.69 | 2.69 |