Assay Report Card

Basic Information

ID: ALA5233090

Type: Binding

Description: Irreversible inhibition of human recombinant tissue transglutaminase expressed in Escherichia coli using Cbz-Glu-(gamma-p-nitrophenylester)Gly (AL5) as substrate assessed as substrate hydrolysis by measuring Kinact/Ki ratio by linear regression analysis

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
359.471.181.18
373.501.571.57
393.921.741.74
381.901.231.23
357.450.620.62
373.460.290.29
377.461.471.47
427.472.112.11
399.891.521.52
438.371.901.90
347.481.981.98