Assay Report Card

Basic Information

ID: ALA5238046

Type: Binding

Description: Protac activity at BRD4/VHL E3 ligase in human MDA-MB-231 cells assessed as decrease in BRD4 expression at 1 uM incubated for 4 hrs by Western blot analysis

Organism: Homo sapiens

Cell type: MDA-MB-231

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
785.283.683.68
771.263.293.29
799.314.074.07
868.424.104.10