Assay Report Card

Basic Information

ID: ALA5238048

Type: Binding

Description: Protac activity at BRD4/VHL E3 ligase in human MDA-MB-231 cells assessed as decrease in BRD4 expression at 1 uM incubated for 16 hrs by Western blot analysis

Organism: Homo sapiens

Cell type: MDA-MB-231

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
801.282.922.92
785.283.683.68
771.263.293.29
845.332.942.94
799.314.074.07
786.274.114.11
840.363.323.32
854.393.713.71
868.424.104.10