Assay Report Card

Basic Information

ID: ALA5238055

Type: Binding

Description: Protac activity at BRD4/VHL E3 ligase in human MDA-MB-231 cells assessed as decrease in BRD4 expression at 1 uM incubated for 4 to 24 hrs by Western blot analysis

Organism: Homo sapiens

Cell type: MDA-MB-231

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1002.66
941.585.015.01
996.664.694.69
1024.71