Basic Information
ID: ALA5238222
Type: Binding
Description: Inhibition of CDK7 (unknown origin) assessed as phosphorylation of ULight 4EBP1 peptide substrate measured after 2 hrs by FRET-based LANCE Ultra KinSelect assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5238222
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 566.07 | 6.33 | 6.33 |
| 463.54 | 5.07 | 5.07 |
| 532.60 | 5.02 | 5.02 |
| 373.42 | 3.28 | 3.28 |
| 476.54 | 4.39 | 4.39 |
| 314.35 | 3.88 | 3.88 |
| 518.58 | 5.15 | 5.15 |
| 373.42 | 3.21 | 3.21 |
| 545.60 | 4.51 | 4.51 |
| 449.51 | 5.02 | 5.02 |
| 476.54 | 4.39 | 4.39 |
| 531.58 | 4.64 | 4.64 |
| 371.40 | 3.24 | 3.24 |
| 463.54 | 5.07 | 5.07 |
| 449.51 | 5.02 | 5.02 |
| 477.57 | 5.14 | 5.14 |
| 477.57 | 5.14 | 5.14 |
| 462.56 | 5.03 | 5.03 |
| 463.54 | 4.83 | 4.83 |
| 518.58 | 5.15 | 5.15 |
| 344.37 | 3.89 | 3.89 |
| 449.51 | 4.96 | 4.96 |
| 372.43 | 3.25 | 3.25 |
| 462.51 | 4.52 | 4.52 |
| 518.58 | 5.15 | 5.15 |
| 386.42 | 2.77 | 2.77 |
| 328.38 | 4.19 | 4.19 |
| 463.54 | 4.83 | 4.83 |
| 449.51 | 4.96 | 4.96 |
| 330.35 | 3.58 | 3.58 |