Assay Report Card

Basic Information

ID: ALA5238560

Type: Binding

Description: Antagonist activity at glucocorticoid receptor (unknown origin) transfected in human HeLa cells assessed as inhibition of dexamethasone-induced transactivation of receptor at 10 uM incubated for 18 hrs by firefly luciferase assay

Organism: Homo sapiens

Cell type: HeLa

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
392.471.901.90
591.495.765.76
505.425.705.70
680.405.985.98
446.914.344.34
538.986.076.07
612.604.274.27
414.533.803.80
426.522.382.38
477.015.115.11
630.796.216.21
531.035.075.07
484.885.355.35
527.096.396.39
412.473.683.68
572.624.204.20
638.684.034.03
471.974.454.45
427.443.583.58
634.827.057.05
424.483.613.61
529.014.844.84
503.005.505.50
440.524.304.30
450.444.694.69
407.453.553.55
456.614.974.97
400.433.813.81
477.035.325.32
460.944.644.64
432.504.834.83
425.472.772.77
534.664.584.58
475.574.894.89
436.534.554.55
521.046.206.20
582.664.474.47
550.665.075.07
461.884.244.24
438.555.025.02
412.473.683.68
524.583.253.25
658.606.496.49
460.944.644.64
472.953.843.84
522.604.464.46
550.664.744.74
458.545.345.34
501.005.065.06
674.807.797.79
438.554.974.97
382.443.673.67
482.623.943.94
558.584.744.74
634.786.896.89
388.473.733.73
485.015.365.36
450.564.714.71