Assay Report Card

Basic Information

ID: ALA5240529

Type: Binding

Description: Protac activity at CRBN/BRD4 in human MM1.S cells assessed as induction of BRD4 protein degradation by measuring residual activity at 0.6 uM incubated for 3 hrs by Western blot analysis relative to control

Organism: Homo sapiens

Cell type: MM1.S

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
860.405.535.53
861.385.505.50
847.355.115.11