Assay Report Card

Basic Information

ID: ALA5240545

Type: Binding

Description: Protac activity at CRBN/BRD4 in human MV4-11 cells assessed as induction of BRD4 protein degradation by measuring residual activity at 0.003 uM incubated for 3 hrs by Western blot analysis relative to control

Organism: Homo sapiens

Cell type: MV4-11

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
798.334.114.11
875.415.895.89