Assay Report Card

Basic Information

ID: ALA5246745

Type: Binding

Description: Inhibition of N-terminal GST-fused human wild type LRRK2 using fluorescein-labeled LRRKtide as substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by TR-FRET assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
353.350.010.01
324.351.221.22
324.351.301.30
409.450.610.61
500.572.552.55
350.391.731.73
389.221.671.67
473.501.211.21
354.370.780.78
367.370.960.96
353.340.480.48
324.351.471.47
354.370.780.78
472.511.811.81
296.290.520.52
387.411.971.97
310.320.910.91
338.381.781.78
338.381.781.78
395.431.651.65
414.473.313.31
323.361.831.83
352.401.961.96
486.542.372.37
326.320.210.21
338.330.830.83
324.351.301.30
465.501.231.23
325.330.530.53
324.350.990.99
372.392.612.61
401.432.532.53
324.350.990.99
339.360.840.84
429.442.162.16
426.442.462.46
338.381.651.65
324.351.471.47
486.542.372.37
310.320.910.91