Basic Information
ID: ALA5251370
Type: Binding
Description: Inhibition of recombinant human DYRK1B expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis
Organism: Homo sapiens
Cell type: Sf9
Activity Charts
Bioactivity
Activity Types for Assay ALA5251370
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 212.25 | 3.03 | 3.03 |
| 368.39 | 3.37 | 3.37 |
| 505.46 | 4.18 | 4.18 |
| 458.38 | 2.23 | 2.23 |
| 228.29 | 3.42 | 3.42 |
| 260.20 | 1.77 | 1.77 |
| 452.29 | 2.97 | 2.97 |
| 245.24 | 0.54 | 0.54 |
| 464.47 | 0.27 | 0.27 |
| 570.65 | 5.91 | 5.91 |
| 320.40 | 2.59 | 2.59 |
| 323.37 | 2.98 | 2.98 |
| 349.78 | 4.88 | 4.88 |
| 235.31 | 2.75 | 2.75 |
| 338.19 | 3.48 | 3.48 |
| 388.48 | 3.88 | 3.88 |
| 210.24 | 2.92 | 2.92 |
| 307.31 | 2.35 | 2.35 |
| 362.46 | 4.65 | 4.65 |
| 298.30 | 3.56 | 3.56 |
| 194.24 | 3.23 | 3.23 |
| 506.61 | 4.94 | 4.94 |
| 429.53 | 3.53 | 3.53 |
| 388.16 | 4.17 | 4.17 |
| 383.41 | 4.10 | 4.10 |
| 271.71 | 3.38 | 3.38 |
| 347.54 | ||
| 320.32 | 4.45 | 4.45 |
| 505.56 | 6.35 | 6.35 |
| 282.35 | 2.55 | 2.55 |
| 316.37 | 3.26 | 3.26 |
| 494.53 | 3.60 | 3.60 |
| 352.40 | 4.96 | 4.96 |
| 487.91 | 5.40 | 5.40 |
| 427.51 | 3.03 | 3.03 |
| 471.60 | 6.57 | 6.57 |
| 240.27 | 1.25 | 1.25 |
| 319.32 | 3.41 | 3.41 |
| 322.29 | 2.53 | 2.53 |
| 401.28 | 5.02 | 5.02 |
| 486.43 | 3.61 | 3.61 |
| 378.50 | 3.68 | 3.68 |
| 468.44 | 3.47 | 3.47 |
| 328.44 | 3.85 | 3.85 |
| 476.63 | 3.14 | 3.14 |
| 546.59 | 4.70 | 4.70 |
| 311.34 | 2.31 | 2.31 |
| 537.40 | 5.67 | 5.67 |
| 340.45 | 3.44 | 3.44 |
| 335.39 | 4.02 | 4.02 |
| 413.50 | 2.25 | 2.25 |
| 449.56 | 4.55 | 4.55 |
| 384.50 | 3.60 | 3.60 |
| 481.60 | 3.87 | 3.87 |
| 299.36 | 3.33 | 3.33 |
| 391.52 | 3.94 | 3.94 |