ID: ALA5251379
Type: Binding
Description: Inhibition of recombinant human DYRK1A expressed in Escherichia coli using DYRKtide peptide as substrate incubated for 110 mins in presence of ATP by non-radioactive ADP-Glo luminescence microplate reader assay
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA5251379
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
212.25 | 3.03 | 3.03 |
368.39 | 3.37 | 3.37 |
458.38 | 2.23 | 2.23 |
452.29 | 2.97 | 2.97 |
349.78 | 4.88 | 4.88 |
338.19 | 3.48 | 3.48 |
388.48 | 3.88 | 3.88 |
307.31 | 2.35 | 2.35 |
362.46 | 4.65 | 4.65 |
298.30 | 3.56 | 3.56 |
194.24 | 3.23 | 3.23 |
506.61 | 4.94 | 4.94 |
429.53 | 3.53 | 3.53 |
388.16 | 4.17 | 4.17 |
383.41 | 4.10 | 4.10 |
271.71 | 3.38 | 3.38 |
320.32 | 4.45 | 4.45 |
505.56 | 6.35 | 6.35 |
282.35 | 2.55 | 2.55 |
494.53 | 3.60 | 3.60 |
427.51 | 3.03 | 3.03 |
319.32 | 3.41 | 3.41 |
322.29 | 2.53 | 2.53 |
401.28 | 5.02 | 5.02 |
486.43 | 3.61 | 3.61 |
378.50 | 3.68 | 3.68 |
468.44 | 3.47 | 3.47 |
546.59 | 4.70 | 4.70 |
311.34 | 2.31 | 2.31 |
340.45 | 3.44 | 3.44 |
335.39 | 4.02 | 4.02 |
413.50 | 2.25 | 2.25 |
481.60 | 3.87 | 3.87 |
299.36 | 3.33 | 3.33 |
391.52 | 3.94 | 3.94 |