Assay Report Card

Basic Information

ID: ALA5251703

Type: Binding

Description: Inhibition of human C-terminal his tagged DYRK1A (26 to 490 residues) transfected in HEK293T cells assessed as inhibition of cyclin D1 phosphorylation at 10 uM incubated for 3 hrs by by Western blot analysis

Organism: Homo sapiens

Cell type: HEK293T

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
212.253.033.03
328.173.493.49
349.784.884.88