ID: ALA5251900
Type: Binding
Description: Inhibition of EGFR (unknown origin) preincubated for 1 hrs followed by substrate addition and measured after 1 hrs in the presence of ATP at Km concentration by TR-FRET assay
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA5251900
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
506.01 | 4.88 | 4.88 |
501.59 | 4.23 | 4.23 |
483.57 | 4.06 | 4.06 |
507.54 | 4.50 | 4.50 |
471.56 | 4.22 | 4.22 |
471.56 | 4.22 | 4.22 |
421.55 | 3.36 | 3.36 |
482.80 | 4.39 | 4.39 |
453.54 | 2.76 | 2.76 |
531.61 | 4.24 | 4.24 |
479.61 | 3.96 | 3.96 |
479.58 | 3.32 | 3.32 |
479.58 | 3.11 | 3.11 |
467.57 | 3.01 | 3.01 |
481.60 | 3.40 | 3.40 |
522.83 | 3.85 | 3.85 |
487.56 | 4.07 | 4.07 |
507.64 | 4.11 | 4.11 |
465.58 | 3.65 | 3.65 |
487.56 | 3.93 | 3.93 |
518.41 | 3.21 | 3.21 |
453.54 | 2.76 | 2.76 |
481.60 | 3.57 | 3.57 |
461.52 | 3.50 | 3.50 |
527.25 | 4.50 | 4.50 |
518.41 | 3.21 | 3.21 |
449.51 | 3.19 | 3.19 |
479.58 | 3.32 | 3.32 |
473.96 | 3.10 | 3.10 |