Assay Report Card

Basic Information

ID: ALA5252745

Type: Binding

Description: Inhibition of human recombinant GST-fused VEGFR1 kinase domain transphosphorylation expressed in baculovirus expression system using poly-Glu-Tyr (4:1) as substrate measured after 10 mins in presence of gamma-[33P]-ATP by scintillation counting analysis

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
398.483.333.33
464.915.015.01
371.364.964.96
464.835.555.55
439.395.195.19
424.385.285.28
442.375.415.41
442.375.415.41
424.385.285.28