Basic Information
ID: ALA5252748
Type: Binding
Description: Inhibition of human recombinant GST-fused VEGFR2 kinase domain transphosphorylation expressed in baculovirus expression system using poly-Glu-Tyr (4:1) as substrate measured after 10 mins in presence of gamma-[33P]-ATP by scintillation counting analysis
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5252748
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 398.48 | 3.33 | 3.33 |
| 464.91 | 5.01 | 5.01 |
| 371.36 | 4.96 | 4.96 |
| 464.83 | 5.55 | 5.55 |
| 529.57 | 5.11 | 5.11 |
| 439.39 | 5.19 | 5.19 |
| 424.38 | 5.28 | 5.28 |
| 458.83 | 5.93 | 5.93 |
| 500.41 | 6.01 | 6.01 |
| 522.53 | 5.03 | 5.03 |
| 434.38 | 5.56 | 5.56 |
| 442.37 | 5.41 | 5.41 |
| 481.43 | 5.87 | 5.87 |
| 442.37 | 5.41 | 5.41 |
| 384.44 | 4.82 | 4.82 |
| 424.38 | 5.28 | 5.28 |