Assay Report Card

Basic Information

ID: ALA5254782

Type: Binding

Description: Positive allosteric modulation of rat recombinant GABAA alpha6beta3gamma2 receptor expressed in Xenopus laevis oocytes assessed as maximal efficacy at -80 mV holding potential at 300 nM in presence of GABA EC1 to 1.5 by two-electrode voltage-clamp assay

Organism: Rattus norvegicus

Cell type: Oocyte

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
370.213.593.59