Assay Report Card

Basic Information

ID: ALA5256564

Type: Binding

Description: Inhibition of human furin in human PANC-1 cells assessed as release of fluorescent AMC using Pyr-Arg-Thr-Arg-AMC as substrate preincubated for 10 mins in presence of SFTI-1 then incubation with ligand for 30 mins followed by substrate addition by plate reader analysis

Organism: Homo sapiens

Cell type: PANC-1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1555.99
1584.00
1601.03
1416.83