Basic Information
ID: ALA5258418
Type: Binding
Description: Inhibition of CDK2/Cyclin E1 (unknown origin) assessed as inhibition of substrate peptide phosphorylation using eIF4E-binding protein 1 as peptide substrate incubated for 4 hrs in presence of ATP by Lance Ultra HTRF assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5258418
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 432.31 | 3.60 | 3.60 |
| 356.43 | 2.40 | 2.40 |
| 369.43 | 2.97 | 2.97 |
| 386.46 | 2.68 | 2.68 |
| 402.56 | 3.88 | 3.88 |
| 357.41 | 2.83 | 2.83 |
| 367.45 | 3.73 | 3.73 |
| 420.56 | 4.44 | 4.44 |
| 369.43 | 3.20 | 3.20 |
| 295.32 | 3.31 | 3.31 |
| 370.41 | 1.93 | 1.93 |
| 332.41 | 2.66 | 2.66 |
| 329.40 | 3.32 | 3.32 |
| 344.46 | 2.66 | 2.66 |
| 444.49 | 5.38 | 5.38 |
| 437.32 | 2.97 | 2.97 |
| 357.41 | 2.48 | 2.48 |
| 357.41 | 3.08 | 3.08 |
| 406.47 | 1.59 | 1.59 |
| 355.44 | 3.64 | 3.64 |
| 370.41 | 2.04 | 2.04 |
| 409.94 | 3.65 | 3.65 |
| 405.48 | 2.48 | 2.48 |
| 405.46 | 2.07 | 2.07 |