Basic Information
ID: ALA5259078
Type: Binding
Description: Partial agonist activity at N-terminal FLAG tagged/C-terminal NanoLuc tagged human muscarinic M5 receptor expressed in HEK293T cells using furimazine as substrate assessed as receptor activation at 100 uM preincubated with substrate for 1 min followed by compound addition and measured for 6 mins 27 sec by NanoBRET assay
Organism: Homo sapiens
Cell type: HEK293T
Activity Charts
Bioactivity
Activity Types for Assay ALA5259078
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 664.80 | 4.53 | 4.53 |
| 790.68 | 5.95 | 5.95 |
| 720.91 | 5.95 | 5.95 |
| 650.77 | 4.52 | 4.52 |