Basic Information
ID: ALA5259642
Type: Binding
Description: Competitive binding affinity to Nluc-fused human GPR35 expressed in CHO-K1 cells assessed as inhibition constant using furimazine as substrate incubated for 30 mins followed by substrate addition by in presence of 10-(4-(2-(4-(4-((2,8-dicarboxy-6-hydroxy-10-methylpyrido[3,2-g]quinolin-4-yl)oxy)butyl)-1H-1,2,3-triazol-1-yl)ethoxy)phenyl)-5,5-difluoro-2,7,9-trimethyl-5H-imidazo[1,2-c]pyrrolo[2,1-f][1,3,2]diazaborinin-6-ium-5-uide
Organism: Homo sapiens
Cell type: CHO-K1
Activity Charts
Bioactivity
Activity Types for Assay ALA5259642
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 468.37 | 2.11 | 2.11 |
| 271.28 | 1.50 | 1.50 |
| 388.38 | 4.39 | 4.39 |
| 330.21 | 0.55 | 0.55 |
| 482.58 | 4.66 | 4.66 |
| 395.44 | 2.53 | 2.53 |
| 314.25 | 1.07 | 1.07 |
| 363.94 | 2.72 | 2.72 |
| 354.08 | 1.35 | 1.35 |
| 374.20 | 2.89 | 2.89 |
| 408.32 | 2.97 | 2.97 |