Basic Information
ID: ALA5263178
Type: Binding
Description: Displacement of N-alpha-[methyl-3H]-methylhistamine dihydrochloride from Sprague-Dawley rat brain membrane histamine H3 receptor assessed as inhibition constant incubated for 30 mins by liquid scintillation counting analysis
Organism: Rattus norvegicus
Strain: Sprague-Dawley
Tissue: Brain
Subcellular Fraction: Membrane
Activity Charts
Bioactivity
Activity Types for Assay ALA5263178
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 292.45 | 2.80 | 2.80 |
| 295.85 | 4.17 | 4.17 |
| 436.68 | 5.87 | 5.87 |
| 436.68 | 5.87 | 5.87 |
| 450.71 | 6.26 | 6.26 |
| 451.05 | 6.63 | 6.63 |
| 450.71 | 6.26 | 6.26 |
| 430.68 | 5.11 | 5.11 |
| 465.68 | 4.21 | 4.21 |
| 416.61 | 5.98 | 5.98 |
| 493.74 | 4.97 | 4.97 |
| 416.61 | 5.98 | 5.98 |
| 450.71 | 6.12 | 6.12 |
| 466.71 | 5.23 | 5.23 |
| 416.61 | 5.98 | 5.98 |
| 492.75 | 6.08 | 6.08 |
| 422.66 | 5.48 | 5.48 |
| 450.71 | 6.26 | 6.26 |
| 450.71 | 6.26 | 6.26 |
| 452.68 | 4.84 | 4.84 |
| 454.74 | 6.28 | 6.28 |
| 464.74 | 6.65 | 6.65 |