Basic Information
ID: ALA5264188
Type: Binding
Description: Displacement of [3H]GX-545 from human Nav1.7 alpha subunit expressed in HEK293 cells co-expressing beta1 subunit by liquid scintillation counting analysis
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA5264188
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 415.91 | 3.76 | 3.76 |
| 399.46 | 3.25 | 3.25 |
| 335.78 | 2.35 | 2.35 |
| 433.90 | 3.86 | 3.86 |
| 397.92 | 3.62 | 3.62 |
| 431.91 | 2.88 | 2.88 |
| 377.87 | 3.52 | 3.52 |
| 409.52 | 3.67 | 3.67 |
| 421.53 | 3.99 | 3.99 |
| 432.37 | 4.28 | 4.28 |
| 349.81 | 2.74 | 2.74 |
| 349.81 | 2.88 | 2.88 |
| 451.89 | 4.01 | 4.01 |
| 457.51 | 4.23 | 4.23 |
| 395.50 | 3.42 | 3.42 |
| 405.44 | 3.60 | 3.60 |
| 469.88 | 4.04 | 4.04 |
| 431.48 | 4.13 | 4.13 |
| 449.49 | 3.61 | 3.61 |
| 445.50 | 4.52 | 4.52 |
| 435.56 | 4.66 | 4.66 |
| 477.52 | 5.06 | 5.06 |
| 363.84 | 3.13 | 3.13 |
| 369.46 | 3.35 | 3.35 |
| 365.81 | 1.97 | 1.97 |
| 459.53 | 4.91 | 4.91 |
| 423.55 | 4.23 | 4.23 |