Assay Report Card

Basic Information

ID: ALA5264645

Type: Binding

Description: Protac activity at VHL/AR in AR-positive human LNCaP cells assessed as induction of androgen receptor degradation at 10 uM incubated for 6 hrs by Western blot analysis (Rvb = 0%)

Organism: Homo sapiens

Cell type: LNCaP

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
464.443.993.99
1034.73
1129.84
1129.84
1073.28
1061.28
991.157.557.55
935.045.995.99
1125.31
949.076.386.38
1023.14
1045.23
977.127.167.16
963.096.776.77
1059.25