Basic Information
ID: ALA5265513
Type: Binding
Description: Inhibition of human TRPM8 expressed in HEK293 cells assessed as reduction in cold stimulated Ca2+ efflux preincubated for 5 mins followed by cold stimulation and measured for 3 mins
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA5265513
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 251.28 | 3.25 | 3.25 |
| 291.31 | 2.33 | 2.33 |
| 294.31 | 2.43 | 2.43 |
| 292.32 | 2.00 | 2.00 |
| 289.32 | 1.89 | 1.89 |