Assay Report Card

Basic Information

ID: ALA636450

Type: Binding

Description: Binding affinity at human Adenosine A2B receptor expressed in HEK293 cells, using [125I]ABOPX as radioligand

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
336.33-0.13-0.13
282.301.281.28
299.330.690.69
300.270.330.33
300.270.330.33
284.321.591.59
286.290.640.64
301.260.540.54
194.19-1.03-1.03
354.453.263.26
278.361.591.59
194.19-0.18-0.18
278.310.190.19
246.270.270.27
266.26-1.00-1.00
270.290.480.48
208.22-0.07-0.07
232.240.260.26
194.19-0.56-0.56
208.220.000.00
218.22-0.93-0.93
224.22-1.57-1.57
220.23-0.38-0.38
242.67-0.33-0.33
218.22-0.93-0.93
272.260.330.33
386.411.841.84
262.311.481.48
344.371.781.78
376.843.043.04
344.371.781.78
194.19-0.18-0.18
256.260.630.63
236.270.710.71
256.260.470.47
204.19-0.94-0.94
270.720.450.45
256.690.060.06
344.801.991.99
296.331.291.29
284.321.061.06
270.290.670.67
369.432.332.33
208.220.210.21
219.20-1.04-1.04
223.24-1.61-1.61
219.20-1.04-1.04
256.260.660.66
220.230.530.53
218.22-0.93-0.93
236.23-0.98-0.98
374.873.093.09
266.26-1.00-1.00
320.443.053.05
238.20-1.48-1.48
192.18-0.40-0.40
190.16-0.95-0.95
346.260.440.44
224.22-0.96-0.96
238.20-1.48-1.48
374.401.791.79
348.352.652.65
314.351.161.16
344.371.781.78
236.270.710.71
312.372.372.37
358.402.092.09
402.411.541.54
304.392.362.36
180.17-1.04-1.04