Assay Report Card

Basic Information

ID: ALA636669

Type: Binding

Description: Binding affinity against adenosine A1 receptor in rat brain membrane preparations using N6-[3H]cyclohexyladenosine as radioligand, PCY = log (100000/IC50).

Tissue: Brain

Subcellular Fraction: Membrane

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
336.33-0.13-0.13
290.711.281.28
271.280.210.21
316.320.640.64
270.290.940.94
305.730.860.86
257.250.020.02
271.280.210.21
271.280.210.21
316.320.640.64
286.290.640.64
325.151.931.93
316.320.640.64
286.290.640.64
301.260.540.54
301.260.540.54
289.732.282.28
256.260.630.63
270.290.550.55
300.322.062.06
300.322.062.06
241.251.441.44
254.292.532.53
270.292.052.05
300.322.062.06
309.163.353.35
270.292.052.05
270.291.111.11
257.250.020.02
241.251.441.44
255.281.631.63
285.261.951.95
164.170.380.38
254.291.971.97
254.292.352.35
285.261.951.95
240.272.042.04
320.331.291.29
255.281.631.63
274.712.702.70
255.281.631.63
180.17-1.04-1.04