Assay Report Card

Basic Information

ID: ALA651925

Type: Binding

Description: Binding affinity of compound (10 uM) towards H121A/T292A receptor variant (double mutant CCR2 receptor) using radioligand [125I]MCP-1 in HEK 293 cells

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
531.146.786.78
500.476.366.36
480.656.636.63