Basic Information
ID: ALA653418
Type: Binding
Description: Inhibition specific binding of [3H]BK (1.0 nM) to human Bradykinin receptor B2 which was expressed in CHO (Chinese hamster ovary) cells by 50%.
Cell type: CHO
Activity Charts
Bioactivity
Activity Types for Assay ALA653418
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 608.53 | 5.40 | 5.40 |
| 594.50 | 6.09 | 6.09 |
| 594.50 | 4.92 | 4.92 |
| 581.46 | 5.17 | 5.17 |
| 592.48 | 4.98 | 4.98 |
| 592.48 | 4.98 | 4.98 |
| 583.69 | 4.32 | 4.32 |
| 569.66 | 3.93 | 3.93 |
| 610.50 | 4.62 | 4.62 |
| 582.71 | 3.99 | 3.99 |
| 568.68 | 3.96 | 3.96 |
| 585.73 | 4.64 | 4.64 |
| 581.67 | 4.12 | 4.12 |
| 625.73 | 4.03 | 4.03 |
| 583.69 | 4.07 | 4.07 |
| 611.49 | 4.61 | 4.61 |
| 618.52 | 5.74 | 5.74 |
| 565.67 | 4.63 | 4.63 |
| 606.51 | 5.32 | 5.32 |
| 653.57 | 7.47 | 7.47 |
| 592.48 | 5.57 | 5.57 |
| 638.56 | 7.18 | 7.18 |
| 654.55 | 6.87 | 6.87 |
| 656.57 | 6.28 | 6.28 |
| 552.64 | 3.68 | 3.68 |
| 551.65 | 4.29 | 4.29 |
| 620.54 | 5.53 | 5.53 |
| 555.46 | 4.57 | 4.57 |
| 570.65 | 3.92 | 3.92 |
| 624.53 | 4.96 | 4.96 |
| 552.64 | 4.28 | 4.28 |
| 577.69 | 5.05 | 5.05 |
| 627.96 | 5.58 | 5.58 |
| 644.99 | 5.17 | 5.17 |
| 628.94 | 4.98 | 4.98 |
| 587.12 | 4.89 | 4.89 |
| 764.93 | 6.26 | 6.26 |
| 627.96 | 6.18 | 6.18 |
| 570.90 | 6.22 | 6.22 |
| 653.99 | 6.35 | 6.35 |
| 709.86 | 5.79 | 5.79 |
| 665.41 | 4.98 | 4.98 |
| 650.61 | 5.05 | 5.05 |
| 608.35 | 5.62 | 5.62 |
| 624.57 | 4.88 | 4.88 |
| 691.44 | 5.74 | 5.74 |
| 695.83 | 5.44 | 5.44 |
| 641.98 | 5.92 | 5.92 |
| 613.16 | 5.66 | 5.66 |
| 628.94 | 5.57 | 5.57 |
| 727.48 | 6.87 | 6.87 |
| 624.57 | 4.29 | 4.29 |
| 727.48 | 6.87 | 6.87 |
| 764.93 | 6.26 | 6.26 |
| 1304.55 |