Assay Report Card

Basic Information

ID: ALA653420

Type: Binding

Description: Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoid carcinoma) which express Bradykinin receptor B2 by 50%.

Cell type: A-431

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
606.315.665.66
605.326.386.38
542.265.175.17
570.315.955.95
618.366.396.39
678.375.665.66
663.366.256.25
635.305.775.77
543.254.574.57
619.305.395.39
606.305.455.45
604.336.006.00
557.283.933.93
641.786.386.38
728.865.455.45
669.796.286.28
695.836.046.04
698.835.785.78
710.845.835.83
626.775.615.61
641.785.755.75
672.755.985.98
657.786.086.08
641.786.386.38
638.786.086.08
709.865.795.79
652.765.955.95
733.284.844.84
695.835.445.44
731.885.455.45
709.866.076.07
747.315.185.18
721.876.216.21
550.674.394.39
627.756.086.08
733.285.445.44
662.206.736.73
1304.55