Basic Information
ID: ALA653424
Type: Binding
Description: In vitro inhibitory activity towards human bradykinin receptor B2 expressed in CHO cells using [3H]BK (1.0 nM) as a radioligand
Cell type: CHO
Activity Charts
Bioactivity
Activity Types for Assay ALA653424
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 591.50 | 5.58 | 5.58 |
| 608.53 | 5.40 | 5.40 |
| 594.50 | 6.09 | 6.09 |
| 594.50 | 4.92 | 4.92 |
| 581.46 | 5.17 | 5.17 |
| 592.48 | 4.98 | 4.98 |
| 592.48 | 4.98 | 4.98 |
| 583.69 | 4.32 | 4.32 |
| 569.66 | 3.93 | 3.93 |
| 610.50 | 4.62 | 4.62 |
| 582.71 | 3.99 | 3.99 |
| 568.68 | 3.96 | 3.96 |
| 585.73 | 4.64 | 4.64 |
| 581.67 | 4.12 | 4.12 |
| 625.73 | 4.03 | 4.03 |
| 583.69 | 4.07 | 4.07 |
| 627.96 | 5.58 | 5.58 |
| 746.06 | 7.05 | 7.05 |
| 757.08 | 7.05 | 7.05 |
| 663.22 | 6.56 | 6.56 |
| 644.99 | 5.17 | 5.17 |
| 779.13 | 8.06 | 8.06 |
| 708.05 | 6.11 | 6.11 |
| 628.94 | 4.98 | 4.98 |
| 587.12 | 4.89 | 4.89 |
| 695.83 | 5.44 | 5.44 |
| 641.98 | 5.92 | 5.92 |
| 709.03 | 5.50 | 5.50 |
| 1304.55 | ||
| 707.49 | 5.65 | 5.65 |
| 721.51 | 5.99 | 5.99 |
| 803.40 | 5.77 | 5.77 |
| 803.40 | 5.77 | 5.77 |
| 825.45 | 7.44 | 7.44 |
| 804.39 | 5.16 | 5.16 |
| 817.43 | 6.11 | 6.11 |