Basic Information
ID: ALA679705
Type: Binding
Description: In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cells
Cell type: Endothelial cell
Activity Charts
Bioactivity
Activity Types for Assay ALA679705
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 563.68 | 5.97 | 5.97 |
| 565.65 | 4.93 | 4.93 |
| 581.65 | 4.63 | 4.63 |
| 550.64 | 5.23 | 5.23 |
| 586.07 | 5.28 | 5.28 |
| 565.65 | 4.93 | 4.93 |
| 581.65 | 4.63 | 4.63 |
| 630.52 | 5.39 | 5.39 |
| 571.75 | 5.58 | 5.58 |
| 646.59 | 5.75 | 5.75 |
| 541.66 | 4.80 | 4.80 |
| 601.75 | 6.36 | 6.36 |
| 552.68 | 4.61 | 4.61 |
| 557.72 | 5.27 | 5.27 |
| 579.75 | 5.77 | 5.77 |
| 625.53 | 5.39 | 5.39 |
| 441.55 | 3.92 | 3.92 |
| 597.72 | 5.35 | 5.35 |
| 610.41 | 5.28 | 5.28 |
| 556.67 | 5.29 | 5.29 |
| 595.70 | 4.94 | 4.94 |
| 567.69 | 5.34 | 5.34 |
| 549.65 | 5.83 | 5.83 |
| 473.55 | 3.75 | 3.75 |
| 572.44 | 4.27 | 4.27 |
| 601.75 | 6.53 | 6.53 |
| 630.52 | 5.39 | 5.39 |
| 487.58 | 4.40 | 4.40 |
| 619.69 | 6.23 | 6.23 |
| 598.52 | 5.56 | 5.56 |
| 565.72 | 5.52 | 5.52 |
| 554.07 | 5.45 | 5.45 |
| 586.14 | 5.87 | 5.87 |
| 601.69 | 5.78 | 5.78 |
| 618.71 | 6.38 | 6.38 |
| 519.63 | 4.80 | 4.80 |
| 593.77 | 6.34 | 6.34 |
| 549.65 | 4.81 | 4.81 |
| 548.44 | 4.32 | 4.32 |
| 592.48 | 5.42 | 5.42 |
| 638.75 | 4.66 | 4.66 |
| 579.68 | 5.32 | 5.32 |
| 551.63 | 4.62 | 4.62 |
| 585.69 | 6.06 | 6.06 |
| 602.47 | 4.28 | 4.28 |
| 551.63 | 4.62 | 4.62 |
| 551.63 | 4.62 | 4.62 |
| 551.63 | 4.62 | 4.62 |
| 581.72 | 5.22 | 5.22 |
| 581.72 | 5.22 | 5.22 |
| 668.31 | 4.87 | 4.87 |
| 621.31 | 5.03 | 5.03 |
| 612.55 | 5.95 | 5.95 |
| 573.61 | 4.20 | 4.20 |
| 568.66 | 4.66 | 4.66 |
| 699.85 | 5.23 | 5.23 |
| 618.71 | 6.38 | 6.38 |
| 619.77 | 6.53 | 6.53 |
| 567.67 | 5.18 | 5.18 |
| 610.49 | 5.42 | 5.42 |
| 761.10 | ||
| 602.51 | 5.39 | 5.39 |
| 614.73 | 5.86 | 5.86 |