Basic Information
ID: ALA753521
Type: Binding
Description: Displacement of 0.5 nM [3H]bremazocine from guinea pig brain membrane opioid receptor kappa with 100 nM DAGO and 100 nM DPDPE
Format: BAO_0000019
Organism: Cavia porcellus
Target: Kappa opioid receptor(ALA3952)
Document: ALA1126090
Displacement of 0.5 nM [3H]bremazocine from guinea pig brain membrane opioid receptor kappa with 100 nM DAGO and 100 nM DPDPE: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA753521
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 327.38 | 1.30 | 1.30 |
| 341.41 | 1.53 | 1.53 |
| 399.49 | 1.74 | 1.74 |
| 399.49 | 1.74 | 1.74 |
| 495.57 | 2.78 | 2.78 |
| 495.57 | 2.78 | 2.78 |
| 441.52 | 2.07 | 2.07 |
| 453.54 | 2.21 | 2.21 |
| 453.54 | 2.21 | 2.21 |
| 343.42 | 1.32 | 1.32 |
| 315.46 | 3.22 | 3.22 |
| 416.54 | 2.07 | 2.07 |