Assay Report Card

Basic Information

ID: ALA816118

Type: Functional

Description: Inhibition of Vesicular glutamate transporter (VGLUT) by the ability to block the uptake of 250 uM of [3,4-3H]-L-glutamate into synaptic vesicles isolated from rat forebrain at a 20 fold excess (5 mM) of inhibitor

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
277.231.651.65
323.303.213.21
277.231.651.65
277.231.651.65
247.211.641.64
233.181.341.34
247.211.641.64
247.211.641.64
261.191.361.36
323.303.213.21
251.622.282.28
235.171.771.77
235.171.771.77
277.231.651.65
275.221.401.40
321.294.054.05
374.973.163.16
217.181.631.63
296.082.392.39
343.082.242.24
286.072.942.94
296.082.392.39
296.082.392.39