Assay Report Card

Basic Information

ID: ALA856223

Type: Binding

Description: Selectivity for thyrotropin releasing hormone receptor 2 measured as ratio of signaling potency (EC50 for expressing CREB-luciferase reporter) towards THR-R1 to that of THR-R2

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
404.47-0.86-0.86
404.47-0.68-0.68
402.46-0.93-0.93
418.50-0.51-0.51
444.540.240.24