Basic Information
ID: ALA872674
Type: Binding
Description: Ability of compound to compete with 50 pM of 5-[125I]iodo-A-85,380 for receptor binding sites in rat brain membranes at room temperature
Format: BAO_0000249
Tissue: Brain
Subcellular Fraction: Brain membranes
Target: Neuronal acetylcholine receptor; alpha4/beta2(ALA1907596)
Document: ALA1148305
Ability of compound to compete with 50 pM of 5-[125I]iodo-A-85,380 for receptor binding sites in rat brain membranes at room temperature: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA872674
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 208.69 | 2.34 | 2.34 |
| 182.20 | 0.96 | 0.96 |
| 398.66 | 3.94 | 3.94 |
| 394.70 | 4.19 | 4.19 |
| 333.79 | 3.57 | 3.57 |
| 380.67 | 3.80 | 3.80 |
| 198.65 | 1.48 | 1.48 |
| 289.77 | 2.93 | 2.93 |
| 259.28 | 2.02 | 2.02 |
| 320.19 | 2.65 | 2.65 |
| 367.19 | 2.49 | 2.49 |
| 310.18 | 3.19 | 3.19 |
| 293.73 | 2.68 | 2.68 |
| 275.74 | 2.54 | 2.54 |
| 301.78 | 3.04 | 3.04 |
| 293.73 | 2.68 | 2.68 |
| 319.77 | 3.18 | 3.18 |
| 295.73 | 1.29 | 1.29 |
| 354.64 | 3.30 | 3.30 |
| 368.66 | 3.69 | 3.69 |
| 307.76 | 3.07 | 3.07 |
| 372.63 | 3.44 | 3.44 |
| 354.64 | 3.30 | 3.30 |