Basic Information
ID: ALA878164
Type: Binding
Description: In vitro inhibition of endothelin binding to Endothelin B receptor in rat cerebellum was measured using 125-I labelled ET-1 competition assay; No measurable affinity
Tissue: Cerebellum
Activity Charts
Bioactivity
Activity Types for Assay ALA878164
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 492.45 | 4.22 | 4.22 |
| 492.45 | 4.52 | 4.52 |
| 420.39 | 4.29 | 4.29 |
| 452.43 | 3.87 | 3.87 |
| 380.34 | 3.98 | 3.98 |
| 422.40 | 3.86 | 3.86 |
| 362.35 | 3.84 | 3.84 |
| 352.39 | 2.86 | 2.86 |