Basic Information
ID: ALA884701
Type: Binding
Description: Affinity against human calcitonin gene related peptide receptor (1 uM) expressed in SK-N-MC cells using [125I]-CGRP as radioligand after 180 minutes of incubation at pH 7.40
Organism: Homo sapiens
Cell type: SK-N-MC
Activity Charts
Bioactivity
Activity Types for Assay ALA884701
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 747.53 | 4.35 | 4.35 |
| 789.57 | 3.74 | 3.74 |
| 789.57 | 3.74 | 3.74 |
| 830.62 | 3.73 | 3.73 |
| 829.64 | 4.78 | 4.78 |
| 856.62 | 4.14 | 4.14 |
| 857.65 | 3.95 | 3.95 |
| 855.63 | 4.29 | 4.29 |
| 869.66 | 4.41 | 4.41 |
| 881.67 | 4.80 | 4.80 |
| 716.51 | 4.94 | 4.94 |
| 716.51 | 4.94 | 4.94 |
| 716.51 | 4.94 | 4.94 |
| 687.48 | 5.10 | 5.10 |
| 756.58 | 4.81 | 4.81 |
| 680.49 | 2.89 | 2.89 |
| 757.57 | 4.20 | 4.20 |
| 701.50 | 4.43 | 4.43 |
| 716.51 | 4.94 | 4.94 |
| 715.53 | 4.82 | 4.82 |