Assay Report Card

Basic Information

ID: ALA927819

Type: Binding

Description: Activity at human recombinant Nav 1.8 channel expressed in HEK293 cells in inactivated state with prepulse voltage of -40 mV assessed as blockade of TTx-resistant sodium current at 0.03 uM

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
311.775.165.16
302.334.384.38
335.795.255.25
366.855.235.23