Basic Information
ID: ALA957999
Type: Binding
Description: Inhibition of human recombinant 17beta-HSD1 expressed in HEK293 cell lysate assessed as conversion of radiolabeled estrone to estradiol
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA957999
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 270.24 | 2.58 | 2.58 |
| 270.24 | 2.58 | 2.58 |
| 254.24 | 2.87 | 2.87 |
| 302.24 | 1.99 | 1.99 |
| 272.26 | 2.51 | 2.51 |
| 224.26 | 3.39 | 3.39 |
| 254.24 | 2.87 | 2.87 |
| 238.24 | 3.17 | 3.17 |
| 222.24 | 3.46 | 3.46 |
| 286.24 | 2.28 | 2.28 |
| 518.56 | 6.38 | 6.38 |
| 240.26 | 3.10 | 3.10 |
| 240.26 | 3.10 | 3.10 |
| 284.27 | 2.88 | 2.88 |
| 240.26 | 3.10 | 3.10 |
| 406.93 | 3.69 | 3.69 |
| 677.84 | 4.54 | 4.54 |
| 487.75 | 6.66 | 6.66 |
| 470.69 | 6.41 | 6.41 |
| 302.28 | 2.52 | 2.52 |
| 446.59 | 4.71 | 4.71 |
| 508.62 | 6.62 | 6.62 |
| 384.89 | 4.41 | 4.41 |
| 443.10 | 3.47 | 3.47 |
| 528.20 | 3.94 | 3.94 |
| 476.58 | 4.86 | 4.86 |
| 439.52 | 4.19 | 4.19 |
| 497.46 | 3.85 | 3.85 |
| 492.62 | 5.57 | 5.57 |
| 356.51 | 4.81 | 4.81 |
| 443.27 | 6.12 | 6.12 |
| 454.64 | 4.73 | 4.73 |
| 382.47 | 2.22 | 2.22 |
| 420.51 | 5.70 | 5.70 |
| 390.53 | 4.77 | 4.77 |