Assay Report Card

Basic Information

ID: ALA962457

Type: Binding

Description: Inhibition of human 17beta-HSD5 expressed in HEK293 cells assessed as enzyme-mediated transformation of [14C]-4-androstene-3,17-dione in to [14C]-testosterone at 3 uM after 18 hrs

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
286.424.094.09
416.584.854.85
342.484.594.59
358.483.853.85
328.454.124.12
326.444.324.32
340.464.714.71
354.495.105.10
382.545.745.74
398.504.114.11
338.454.494.49
338.495.255.25
352.525.645.64
344.504.674.67
400.565.185.18
326.444.324.32
342.484.774.77
354.494.964.96
368.525.355.35
354.494.964.96
380.535.525.52
312.413.793.79
326.444.184.18
340.464.574.57
326.444.184.18
324.465.015.01