Assay Report Card

Basic Information

ID: ALA972639

Type: Functional

Description: Antagonist activity at full length human VDR expressed in HEK293 cells overexpressing mouse osteopontin vitamin D-responsive element assessed as inhibition of 1,25-(OH)2D3-induced transcriptional activation after 16 hrs by dual luciferase reporter gene assay

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
430.675.955.95
430.675.955.95
472.756.986.98
472.756.986.98