Basic Information
ID: ALA983035
Type: Binding
Description: Inhibition of human PHD2 assessed as hydroxylation of Pro564 in human HIF-1alpha by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA983035
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 356.38 | 0.32 | 0.32 |
| 368.44 | 1.66 | 1.66 |
| 384.44 | 0.79 | 0.79 |
| 340.38 | 1.18 | 1.18 |
| 370.41 | 0.88 | 0.88 |
| 390.83 | 0.97 | 0.97 |
| 390.83 | 0.97 | 0.97 |
| 390.83 | 0.97 | 0.97 |
| 406.44 | 1.47 | 1.47 |
| 384.44 | 1.05 | 1.05 |
| 370.41 | 0.62 | 0.62 |
| 370.41 | 0.71 | 0.71 |
| 324.38 | 1.63 | 1.63 |
| 432.48 | 1.98 | 1.98 |
| 370.41 | 0.46 | 0.46 |
| 426.52 | 1.75 | 1.75 |
| 308.31 | 0.92 | 0.92 |
| 307.33 | 0.95 | 0.95 |
| 306.34 | 1.47 | 1.47 |
| 294.31 | -1.11 | -1.11 |
| 370.41 | 0.62 | 0.62 |
| 412.49 | 1.61 | 1.61 |