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ID: ALA1130611

Journal: Bioorg Med Chem Lett

Title: Synthesis and antibacterial activity of 2-alkoxy penems.

Authors: Afonso A, Hon F, Fett N, Weinstein J, Ganguly AK, Naples L, Hare RS, Miller GH.

Abstract: The phosphite mediated Oxalimide cyclization reaction was extended to 4-dithiocarbonates of N-oxalyl-2-azetidinones to synthesize 2-alkoxy penems 3. In general, the in vitro antibacterial potency of compounds 3 was weak compared to the highly potent 2-alkylthiopenems 2.

CiteXplore: 9873624

DOI: 10.1016/s0960-894x(98)00502-2