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ID: ALA1130788

Journal: Bioorg Med Chem Lett

Title: Synthesis and antitumor activity of leinamycin derivatives: modifications of C-8 hydroxy and C-9 keto groups.

Authors: Kanda Y, Ashizawa T, Saitoh Y, Saito H, Gomi K, Okabe M.

Abstract: A series of leinamycin derivatives were synthesized and evaluated for antitumor activity. Modifications at C-8 and C-9 positions revealed a broad structure-activity relationship in vitro and some derivatives showed potent antiproliferative activity against HeLa S3 cells.

CiteXplore: 9871510

DOI: 10.1016/s0960-894x(98)00133-4