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ID: ALA1130941

Journal: Bioorg Med Chem Lett

Title: Comparison of the intrinsic kinase activity and substrate specificity of c-Abl and Bcr-Abl.

Authors: Wu JJ, Phan H, Lam KS.

Abstract: We studied the intrinsic tyrosine kinase activity and substrate specificity of c-Abl and Bcr-Abl protein tyrosine kinases (PTKs) using the peptide substrates discovered from a synthetic combinatorial peptide library. Our data indicate that the phosphorylation of these peptides by Bcr-Abl was consistently stronger than that by c-Abl. Bcr-Abl also showed substrate preference towards those peptides with one or more positive charges.

CiteXplore: 9873528

DOI: 10.1016/s0960-894x(98)00413-2