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ID: ALA1131681

Journal: Bioorg Med Chem Lett

Title: Thiazolo[4,5-d]pyrimidine thiones and -ones as corticotropin-releasing hormone (CRH-R1) receptor antagonists.

Authors: Beck JP, Curry MA, Chorvat RJ, Fitzgerald LW, Gilligan PJ, Zaczek R, Trainor GL.

Abstract: A series of thiazolo[4,5-d]pyrimidine thiones and -ones was prepared and discovered to have good binding affinity to the CRH-R1 receptor, thus showing promise as a new class of potential anxiolytics and/or antidepressants.

CiteXplore: 10328310

DOI: 10.1016/s0960-894x(99)00159-6