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ID: ALA1132668

Journal: Bioorg Med Chem Lett

Title: The design of potent and selective inhibitors of thrombin utilizing a piperazinedione template: part 1.

Authors: Cody WL, Cai C, Doherty AM, Edmunds JJ, He JX, Narasimhan LS, Plummer JS, Rapundalo ST, Rubin JR, Van Huis CA, St-Denis Y, Winocour PD, Siddiqui MA.

Abstract: Utilizing X-ray crystallography and molecular modeling, highly potent and selective peptidomimetic thrombin inhibitors have been designed containing a rigid piperazinedione template. The synthesis and biological activity of these compounds will be described.

CiteXplore: 10498196

DOI: 10.1016/s0960-894x(99)00418-7