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ID: ALA1132799

Journal: Bioorg Med Chem Lett

Title: Hybridization of non-sulfonylurea insulin secretagogue and thiazolidinedione-derived insulin sensitizer.

Authors: Kitajima H, Nakamura M, Tamakawa H, Goto N.

Abstract: Hybrid compounds of non-sulfonylurea insulinotropic agents and thiazolidinedione-derived insulin-sensitizing agents were designed and synthesized. The benzylidenesuccinic acid derivative 24 was equal both to nateglinide in potency of insulin-releasing activity and to pioglitazone in insulin-sensitizing activity.

CiteXplore: 11078199

DOI: 10.1016/s0960-894x(00)00491-1