Document Report Card
Basic Information
ID: ALA1133125
Journal: Bioorg Med Chem Lett
Title: A sigma-1 receptor selective analogue of BD1008. A potential substitute for (+)-opioids in sigma receptor binding assays.
Authors: Maeda DY, Williams W, Bowen WD, Coop A.
Abstract: A simple, achiral monoamine sigma-1 (sigma1) receptor selective ligand (sigma2Ki/sigma1Ki>2000) is described, which could replace the chiral (+)-pentazocine or dextrallorphan as a sigma1 masking agent in sigma2 binding assays.
CiteXplore: 10636233